IRAK-4 protein kinase inhibitor 2

CAS No. 301675-24-1

IRAK-4 protein kinase inhibitor 2( —— )

Catalog No. M28816 CAS No. 301675-24-1

IRAK-4 protein kinase inhibitor 2 is a potent interleukin-1 receptor-associated kinase-4 (IRAK-4) inhibitor(IC50 = 4 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
10MG 35 Get Quote
25MG 56 Get Quote
50MG 82 Get Quote
100MG 120 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    IRAK-4 protein kinase inhibitor 2
  • Note
    Research use only, not for human use.
  • Brief Description
    IRAK-4 protein kinase inhibitor 2 is a potent interleukin-1 receptor-associated kinase-4 (IRAK-4) inhibitor(IC50 = 4 μM).
  • Description
    IRAK-4 protein kinase inhibitor 2 is a potent interleukin-1 receptor-associated kinase-4 (IRAK-4) inhibitor(IC50 = 4 μM).(In Vitro):IRAK-4 protein kinase inhibitor 2 inhibited IRAK-1 (IC50 <10 μM) as well.
  • In Vitro
    IRAK-4 protein kinase inhibitor 2 (compound 1) also inhibits IRAK-1, with an IC50 of <10 μM.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Immunology/Inflammation
  • Target
    IRAK
  • Recptor
    α1-adrenoceptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    301675-24-1
  • Formula Weight
    282.259
  • Molecular Formula
    C14H10N4O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 10 mg/mL (35.43 mM)
  • SMILES
    [O-][N+](=O)c1cccc(c1)C(=O)Nc1nc2ccccc2[nH]1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Boschi D, et al. New potential uroselective NO-donor alpha1-antagonists. J Med Chem. 2003 Aug 14;46(17):3762-5.
molnova catalog
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